DPP-4 Inhibitors

Cat.No.	Product Name	Information
S4002	Sitagliptin phosphate monohydrate	Sitagliptin phosphate (MK-0431) is a potent inhibitor of DPP-IV with IC50 of 19 nM in Caco-2 cell extracts.
S1344	Glimepiride	Glimepiride is a medium-to-long acting sulfonylurea anti-diabetic compound with an ED50 of 182 μg/kg.
S1540	Saxagliptin (BMS-477118,Onglyza)	Saxagliptin (BMS-477118, Onglyza) is a selective and reversible DPP4 inhibitor with IC50 of 26 nM.
S3031	Linagliptin (BI-1356)	Linagliptin is a highly potent, selective DPP-4 inhibitor with IC50 of 1 nM.
S3033	Vildagliptin (LAF-237)	Vildagliptin (LAF-237) inhibits DPP−4 with IC50 of 2.3 nM.
S2868	Alogliptin (SYR-322)	Alogliptin(SYR-322) is a potent, selective inhibitor of DPP-4 with IC50 of < 10 nM.

Cat.No.	Product Name	Solubility (25°C)
Cat.No.	Product Name	Water	DMSO	Ethanol
S4002	Sitagliptin phosphate monohydrate	101 mg/mL	101 mg/mL	<1 mg/mL
S1344	Glimepiride	<1 mg/mL	11 mg/mL	<1 mg/mL
S1540	Saxagliptin (BMS-477118,Onglyza)	63 mg/mL	63 mg/mL	24 mg/mL
S3031	Linagliptin (BI-1356)	<1 mg/mL	17 mg/mL	1 mg/mL
S3033	Vildagliptin (LAF-237)	60 mg/mL	60 mg/mL	60 mg/mL
S2868	Alogliptin (SYR-322)	2 mg/mL	68 mg/mL	<1 mg/mL

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